-
Casein Kinase Related Products (93)
Related Products (93)
-
dCK1α-2
0 ImagesSynonyms: LC-05-004dCK1α-2 is an orally active CK1α molecular glue degrader that targets p53 pathway-related targets. dCK1α-2 exhibits anti-tumor efficacy in mouse models and can increase the expression of p53-related genes..
-
CSNK1-IN-1
0 ImagesCSNK1-IN-1 is a CSNK1A1 inhibitor. CSNK1-IN-1 has inhibitory activity for CSNK1A1 kinase with IC50 values of 21 μM. CSNK1-IN-1 can be used for the research of proliferative disorders.
-
(R,R)-BMS-986397
0 Images(R,R)-BMS-986397 is a CK1α degrader (DC50 between 0.1-0.5 pM). (R,R)-BMS-986397 can be used in anti-leukemia research.
-
Casein kinase 1δ-IN-8
0 ImagesCasein kinase 1δ-IN-8 (compound 494) is an inhibitor of Casein kinase 1δ, Casein kinase 1δ-IN-8 can be used in the study of neurodegenerative disorders such as Alzheimer's disease.
-
Casein Kinase II Inhibitor IV
0 ImagesCasein Kinase II Inhibitor IV is a potent, ATP-competitive of casein kinase II inhibitor with an IC50 of 9 nM. Casein Kinase II Inhibitor IV ia also a human keratinocytes (NHEK) differentiation inducer.
-
Casein Kinase II Inhibitor IV hydrochloride
0 ImagesCat. No.: HY-111378ACAS No.: 2320347-54-2Casein Kinase II Inhibitor IV Hydrochloride is a small-molecule inducer of epidermal keratinocyte differentiation.
-
LY294002 (Standard)
0 ImagesLY294002 (Standard) is the analytical standard of LY294002. This product is intended for research and analytical applications. LY294002 is a broad-spectrum inhibitor of PI3K with IC50s of 0.5, 0.57, and 0.97 μM for PI3Kα, PI3Kδ and PI3Kβ, respectively. LY294002 also inhibits CK2 with an IC50 of 98 nM. LY294002 is a competitive DNA-PK inhibitor that binds reversibly to the kinase domain of DNA-PK with an IC50 of 1.4?μM. LY294002 is an apoptosis activator.
-
CX-5011 free base
0 ImagesCat. No.: HY-50733CAS No.: 1009821-06-0
-
PF-4800567 hydrochloride
0 ImagesCat. No.: HY-12470ACAS No.: 1391052-28-0PF-4800567 hydrochloride is a potent and selective inhibitor of?casein kinase?1? (CK1?), with an?IC50?of 32 nM, which is greater than 20-fold selectivity over CK1δ (IC50, 711 nM). PF-4800567 hydrochloride is useful in probing unique roles between these two kinases in multiple signaling pathways.
-
Emodin-d4
0 ImagesCat. No.: HY-14393SCAS No.: 132796-52-2Synonyms: Frangula emodin-d4Emodin-d4 is the deuterium labeled Emodin. Emodin (Frangula emodin), an anthraquinone derivative, is an anti-SARS-CoV compound. Emodin blocks the SARS coronavirus spike protein and angiotensin-converting enzyme 2 (ACE2) interaction. Emodin inhibits casein kinase-2 (CK2). Anti-inflammatory and anticancer effects. Emodin is a potent selective 11β-HSD1 inhibitor with the IC50 of 186 and 86 nM for human and mouse 11β-HSD1, respectively. Emodin ameliorates metabolic disorder in diet-induced obese mice.
-
Casein kinase 1δ-IN-20
0 ImagesCat. No.: HY-169690CAS No.: 757224-44-5Casein kinase 1δ-IN-20 (compound 427) is a potent casein kinase 1δ inhibitor. Casein kinase 1δ-IN-20 can be used in the study of neurodegenerative diseases such as Alzheimer's disease.
-
Casein kinase 1δ-IN-21
0 ImagesCat. No.: HY-169692CAS No.: 782457-22-1Casein kinase 1δ-IN-21 (compound 501) is a potent casein kinase 1δ inhibitor. Casein kinase 1δ-IN-21 can be used in the study of neurodegenerative diseases such as Alzheimer's disease.
-
Casein kinase 1δ-IN-26
0 ImagesCat. No.: HY-169709CAS No.: 756857-71-3Casein kinase 1δ-IN-26 (compound 505) is a potent casein kinase 1δ inhibitor. Casein kinase 1δ-IN-26 can be used in the study of neurodegenerative diseases such as Alzheimer's disease.
-
Casein kinase 1δ-IN-13
0 ImagesCat. No.: HY-156913CAS No.: 345616-08-2Casein kinase 1δ-IN-13 (compound 401) is a Casein kinase 1δ inhibitor. Casein kinase 1δ-IN-13 can be used in neurodegenerative disease research.
-
CK2-IN-8
0 ImagesCat. No.: HY-155987CAS No.: 442571-27-9CK2-IN-8 (compound 5c) is a CK2 inhibitor with IC50 >33 μM.
-
Casein kinase 1δ-IN-23
0 ImagesCat. No.: HY-169702CAS No.: 729579-66-2Casein kinase 1δ-IN-23 (compound 423) is a potent casein kinase 1δ inhibitor. Casein kinase 1δ-IN-22 can be used in the study of neurodegenerative diseases such as Alzheimer's disease.
